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Pimobendan

Pembrolimus yana da ilimin chemisches Medikament, das verwendet wird, um leichte, mittlere oder schwere kongesttive Herzinsuffizienz zu behandeln, die durch atrioventrikuläre Klappeninsuffizienz da Myokardhypertrophie bei Hunden verursacht wird.
  • 74150-27-9

  • Saukewa: C19H18N4O2

  • 334.37

  • 640-420-7

samuwa:

Bayanin Samfura

Pimobendan


Bayanin Samfura


Pimobendan (C₂₀H₁₈ N₄O₄) wani zaɓi ne na phosphodiesterase III inhibitor da Calcium sensitizer wanda ake amfani dashi sosai a cikin cututtukan zuciya . An wajabta shi da yawa don magance ciwon zuciya a cikin karnuka , inganta aikin zuciya, rage alamun gazawar zuciya, da haɓaka ingancin rayuwa..

Pimobendan yana da ƙima don tsarin aikin sa na biyu , yana haɗa ingantaccen tasirin inotropic tare da vasodilation , yana mai da shi babban jigon jigon don kula da cututtukan zuciya na canine..




Mabuɗin Gano Samfur


  • Sunan samfur: Pimobendan

  • Synonyms: Vetmedin, Pimobendan Hydrochloride (na hydrochloride gishiri)

  • Chemical Formula: C₂₀H₁₈N₄O₄

  • Lambar CAS: 20335-16-4

  • Nauyin Kwayoyin Halitta: 386.39 g/mol

  • Bayyanar: Fari zuwa kashe-fari crystalline foda

  • Wari: Mara wari

  • Solubility: Dan kadan mai narkewa cikin ruwa; mai narkewa a cikin kwayoyin kaushi kamar methanol da ethanol




Chemical & Jiki Properties


Dukiya Matsakaicin Mahimmancin
Tsafta ≥ 99% (maganin magunguna)
Matsayin narkewa 184-188 ° C
Yawan yawa 1.35 g/cm³
Kwanciyar hankali Barga a ƙarƙashin shawarar ajiya yanayin; kariya daga haske da danshi
Hygroscopicity Non-hygroscopic
Siffar Crystalline foda



Manufacturing & Quality Control


An haɗa Pimobendan ta hanyar haɗakarwar kwayoyin halitta mai matakai da yawa a ƙarƙashin yanayin GMP . Kula da inganci yana tabbatar da:


  • High sinadaran da kuma Pharmaceutical tsarki

  • Ƙananan ragowar kaushi da ƙazanta

  • Yarda da dokokin likitancin dabbobi

Kowane tsari yana jurewa gwajin HPLC, nazarin danshi, da duban bayyanar don tabbatar da aminci da aminci.




Aikace-aikace na Pimobendan


Likitan cututtukan zuciya


  • Ana amfani dashi don sarrafa gazawar zuciya (CHF) a cikin karnuka , musamman rashin isashshen zuciya da cututtukan zuciya valvular..

  • Yana inganta haɓakar zuciya, ƙarar bugun jini, da juriyar motsa jiki.

  • Yana rage alamun asibiti kamar gajiya, tari, da edema.


Binciken Magunguna


  • Aiwatar azaman mahallin bincike a cikin nazarin ilimin halittar zuciya da ci gaban ƙwayoyi.

  • An bincika don tasirin injina akan fahimtar calcium da hana PDE.


Aikace-aikace Formulation


  • An haɗa shi cikin allunan baka na dabbobi, capsules, da haɗe-haɗe.

  • Mai jituwa tare da daidaitattun abubuwan haɓaka don barga da sifofin sashi na rayuwa.




Packaging & Logistics


  • Daidaitaccen Marufi:

    • 100 g, 500 g, 1 kg Pharmaceutical-sa foda a shãfe haske amber HDPE kwantena.

    • Akwai marufi na al'ada akan buƙata


  • Yanayin Ajiya:

    • Ajiye a wuri mai sanyi, bushe, da duhu

    • Rike kwantena a rufe sosai

    • Guji zafin zafi, zafi, da hasken rana kai tsaye




Tsaro & Gudanarwa


  • Karɓa tare da daidaitaccen dakin gwaje-gwaje ko matakan kariya na magunguna

  • A guji shakar foda da doguwar fata

  • Yi amfani da PPE mai dacewa gami da safar hannu, tabarau, da rigar lab

  • Tuntuɓi Takardar Bayanan Tsaro (SDS/MSDS) don cikakken kulawa, ajiya, da umarnin gaggawa




Ka'ida & Takardu


Akwai akan buƙata:

  • COA (Takaddun Takaddun Bincike)

  • SDS / MSDS

  • TDS (Takardar Bayanan Fasaha)

  • Yarda da magunguna na dabbobi da takaddun GMP




Me yasa Zabi Mu Pimobendan?


  • ✔ Tsabtataccen matakin magunguna (≥99%)

  • ✔ Ya dace da kayan aikin likitan dabbobi da aikace-aikacen bincike

  • ✔ Marufi masu sassauƙa da zaɓuɓɓukan wadatar kayayyaki

  • ✔ Takaddun shirye-shiryen fitarwa da tallafi na tsari

  • ✔ Jagorar fasaha don tsarawa da haɓaka sashi




Tambayoyin da ake yawan yi (FAQ)


Q1: Menene Pimobendan ake amfani dashi?


Ana amfani da shi da farko don magance raunin zuciya a cikin karnuka, inganta aikin zuciya da rage alamun CHF.


Q2: Shin Pimobendan yana narkewa a cikin ruwa?


Yana da ɗan narkewa a cikin ruwa amma yana narkewa a cikin kaushi na halitta kamar methanol da ethanol.


Q3: Shin za ku iya samar da takaddun nazari da dokoki?


Ee, COA, SDS, TDS, da takaddun yarda da GMP suna samuwa.


Q4: Menene matsakaicin mafi ƙarancin tsari (MOQ)?


MOQ ya dogara da marufi da buƙatun tsari; don Allah a tuntube mu don cikakkun bayanai.

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