74150-27-9
Saukewa: C19H18N4O2
334.37
640-420-7
| samuwa: | |
|---|---|
Bayanin Samfura
Pimobendan (C₂₀H₁₈ N₄O₄) wani zaɓi ne na phosphodiesterase III inhibitor da Calcium sensitizer wanda ake amfani dashi sosai a cikin cututtukan zuciya . An wajabta shi da yawa don magance ciwon zuciya a cikin karnuka , inganta aikin zuciya, rage alamun gazawar zuciya, da haɓaka ingancin rayuwa..
Pimobendan yana da ƙima don tsarin aikin sa na biyu , yana haɗa ingantaccen tasirin inotropic tare da vasodilation , yana mai da shi babban jigon jigon don kula da cututtukan zuciya na canine..
Sunan samfur: Pimobendan
Synonyms: Vetmedin, Pimobendan Hydrochloride (na hydrochloride gishiri)
Chemical Formula: C₂₀H₁₈N₄O₄
Lambar CAS: 20335-16-4
Nauyin Kwayoyin Halitta: 386.39 g/mol
Bayyanar: Fari zuwa kashe-fari crystalline foda
Wari: Mara wari
Solubility: Dan kadan mai narkewa cikin ruwa; mai narkewa a cikin kwayoyin kaushi kamar methanol da ethanol
| Dukiya | Matsakaicin Mahimmancin |
|---|---|
| Tsafta | ≥ 99% (maganin magunguna) |
| Matsayin narkewa | 184-188 ° C |
| Yawan yawa | 1.35 g/cm³ |
| Kwanciyar hankali | Barga a ƙarƙashin shawarar ajiya yanayin; kariya daga haske da danshi |
| Hygroscopicity | Non-hygroscopic |
| Siffar | Crystalline foda |
An haɗa Pimobendan ta hanyar haɗakarwar kwayoyin halitta mai matakai da yawa a ƙarƙashin yanayin GMP . Kula da inganci yana tabbatar da:
High sinadaran da kuma Pharmaceutical tsarki
Ƙananan ragowar kaushi da ƙazanta
Yarda da dokokin likitancin dabbobi
Kowane tsari yana jurewa gwajin HPLC, nazarin danshi, da duban bayyanar don tabbatar da aminci da aminci.
Ana amfani dashi don sarrafa gazawar zuciya (CHF) a cikin karnuka , musamman rashin isashshen zuciya da cututtukan zuciya valvular..
Yana inganta haɓakar zuciya, ƙarar bugun jini, da juriyar motsa jiki.
Yana rage alamun asibiti kamar gajiya, tari, da edema.
Aiwatar azaman mahallin bincike a cikin nazarin ilimin halittar zuciya da ci gaban ƙwayoyi.
An bincika don tasirin injina akan fahimtar calcium da hana PDE.
An haɗa shi cikin allunan baka na dabbobi, capsules, da haɗe-haɗe.
Mai jituwa tare da daidaitattun abubuwan haɓaka don barga da sifofin sashi na rayuwa.
Daidaitaccen Marufi:
100 g, 500 g, 1 kg Pharmaceutical-sa foda a shãfe haske amber HDPE kwantena.
Akwai marufi na al'ada akan buƙata
Yanayin Ajiya:
Ajiye a wuri mai sanyi, bushe, da duhu
Rike kwantena a rufe sosai
Guji zafin zafi, zafi, da hasken rana kai tsaye
Karɓa tare da daidaitaccen dakin gwaje-gwaje ko matakan kariya na magunguna
A guji shakar foda da doguwar fata
Yi amfani da PPE mai dacewa gami da safar hannu, tabarau, da rigar lab
Tuntuɓi Takardar Bayanan Tsaro (SDS/MSDS) don cikakken kulawa, ajiya, da umarnin gaggawa
Akwai akan buƙata:
COA (Takaddun Takaddun Bincike)
SDS / MSDS
TDS (Takardar Bayanan Fasaha)
Yarda da magunguna na dabbobi da takaddun GMP
✔ Tsabtataccen matakin magunguna (≥99%)
✔ Ya dace da kayan aikin likitan dabbobi da aikace-aikacen bincike
✔ Marufi masu sassauƙa da zaɓuɓɓukan wadatar kayayyaki
✔ Takaddun shirye-shiryen fitarwa da tallafi na tsari
✔ Jagorar fasaha don tsarawa da haɓaka sashi
Q1: Menene Pimobendan ake amfani dashi?
Ana amfani da shi da farko don magance raunin zuciya a cikin karnuka, inganta aikin zuciya da rage alamun CHF.
Q2: Shin Pimobendan yana narkewa a cikin ruwa?
Yana da ɗan narkewa a cikin ruwa amma yana narkewa a cikin kaushi na halitta kamar methanol da ethanol.
Q3: Shin za ku iya samar da takaddun nazari da dokoki?
Ee, COA, SDS, TDS, da takaddun yarda da GMP suna samuwa.
Q4: Menene matsakaicin mafi ƙarancin tsari (MOQ)?
MOQ ya dogara da marufi da buƙatun tsari; don Allah a tuntube mu don cikakkun bayanai.
abun ciki fanko ne!